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Concomitant administration of P-gp inhibitors (see sections ‧ and ‧). en Sirolimus is also a substrate for the multidrug efflux pump, P-glycoprotein (P-gp) located. della P-gp (itraconazolo, claritromicina, telitromicina, eritromicina, amiodarone. new/4134-1-9244.php P450; P-gp, P-glycoprotein NR, not reported * Of absorbed substance # Of ingested. n (%) Aspirin Thienopyridine Amiodarone Digoxin or digitalis preparations. label NOAC If INR was <2.0 thrombin inhibitor or FXa inhibitor was started If. new/5736-1-8240.php O: Other (amiodarone, aprepitant, grapefruit juice, starfruit). Mechanism: Inhibition of digoxin transport by P-glycoprotein resulting in reduced. new/4614-1-4535.php Amiodarone (moderato P-gp inibitore) Verapamil (forte P-gp inibitore). DDI drugdrug interaction P-gp P-glycoprotein. Dec 2011. Disclaimer. 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Class verapamil calcium channel blocker quinidine antiarrhythmic amiodarone antiarrhythmic ketoconazole. As a consequence, carboxylation of the calcification inhibitor Matrix Gla Protein. reduced glutathione (GSH) content, and expression of P-glycoprotein (P-gp). Effects of metabolites and analogs of amiodarone on alveolar macrophages:. In addition, many drugs have the characteristics of both substrates and inhibitors of P-gp and CYP3A (eg, amiodarone, quinidine, ketoconazole, calcium channel. Inhibitory activity of the sulfamate derivatives against steroid sulfatase and carbonic. Keywords: (3 Iodobenzyl)guanidine I 123, Amiodarone, Beta Adrenergic R. Keywords: Bcl-2, Drug Resistance, P-Glycoprotein, Abc Transporter, Erl. concomitant use of strong inhibitors of P-glycoprotein, as quinidine. Edoxaban coadministered with amiodarone increased total exposure by < 50%. 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