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Partial Dopamine Agonism • Aripiprazole (OPC-14597) – High Affinity for D2 and D3 receptors • Works on: – Postsynaptic D2 receptors – Presynaptic. Ziprasidone also has a high affinity for 5HT1A (where it acts as a partial. Unlike other SGAs, aripiprazole is a D2 and D3 receptor partial agonist and it is. Repeated aripiprazole treatment regulates Bdnf, Arc and Npas4 expression under basal. The AMPA receptor potentiator Org 26576 modulates stress-induced. amlodipine cozaar combination PHARMACOLOGICAL PROPERTIES: Aripiprazole is a quinolinone derivative with a high affinity for dopamine D2 and D3 receptors, and serotonin 5-HT1A. Aripiprazole A case report published by Aragona 123 reported the tolerability. Profile of receptor binding, expressed as receptor affinity (Ki) of antipsychotic.
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